AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction

doi:10.1016/j.tetlet.2020.152054

IOCAS-IR > 实验海洋生物学重点实验室

	AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction
	Li, Xiaowei1,3,4 ; Li, Yuxiu 2; Liu, Ruihua 2; Wang, Zemin 2; Li, Xiangqian 2; Shi, Dayong 2,3,4
	2020-06-25
发表期刊	TETRAHEDRON LETTERS
ISSN	0040-4039
卷号	61 期号:26 页码:5
通讯作者	Shi, Dayong([email protected])
摘要	An AcOH-mediated three-component reaction of 2-aminothiophenols, alpha,beta-unsaturated aldehydes, and thiophenols to prepare the high value-added 2-thioalkylbenzothiazoles was developed. The reaction was conducted under metal-free conditions, where oxygen served as the terminal oxidant. In addition, this strategy is tolerant of kinds of functional groups, providing efficient access to a variety of functionalized benzothiazole derivatives in moderate to good yields. What's more, this reaction has complete regioslectivity and provides a powerful method for building complex molecules. (C) 2020 Elsevier Ltd. All rights reserved.
关键词	2-Thioalkylbenzothiazoles Metal-free Aerobic oxidation Multicomponent reaction
DOI	10.1016/j.tetlet.2020.152054
收录类别	SCI
语种	英语
资助项目	Shandong Provincial Natural Science Foundation for Distinguished Young Scholars[JQ201722]; Taishan scholar Youth Project of Shandong province; Qingdao Marine Biomedical Science and Technology Innovation Center Project[2017-CXZX01-1-1]; Qingdao Marine Biomedical Science and Technology Innovation Center Project[2017-CXZX01-3-9]; NSFC-Shandong Joint Fund[U1706213]; National Natural Science Foundation of China[81803344]; China Postdoctoral Science Foundation[2019M662374]; China Postdoctoral Science Foundation[2019M662377]; China Postdoctoral Science Foundation[2019M662378]; National Program for Support of Top-notch Young Professionals; Key research and development plan (soft science) project of Shandong province[2019RKE27018]
WOS研究方向	Chemistry
WOS类目	Chemistry, Organic
WOS记录号	WOS:000540277100014
出版者	PERGAMON-ELSEVIER SCIENCE LTD
引用统计	被引频次：3[WOS] [WOS记录] [WOS相关记录]
文献类型	期刊论文
条目标识符	http://ir.qdio.ac.cn/handle/337002/167673
专题	实验海洋生物学重点实验室
通讯作者	Shi, Dayong
作者单位	1.Chinese Acad Sci, Inst Oceanol, Key Lab Expt Marine Biol, 7 Nanhai Rd, Qingdao 266071, Shandong, Peoples R China 2.Shandong Univ, State Key Lab Microbial Technol, 72 Binhai Rd, Qingdao 266237, Peoples R China 3.Qingdao Natl Lab Marine Sci & Technol, Lab Marine Drugs & Bioprod, Qingdao 266000, Peoples R China 4.Univ Chinese Acad Sci, Beijing 100049, Peoples R China
第一作者单位	中国科学院海洋研究所
推荐引用方式 GB/T 7714	Li, Xiaowei,Li, Yuxiu,Liu, Ruihua,et al. AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction[J]. TETRAHEDRON LETTERS,2020,61(26):5.
APA	Li, Xiaowei,Li, Yuxiu,Liu, Ruihua,Wang, Zemin,Li, Xiangqian,&Shi, Dayong.(2020).AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction.TETRAHEDRON LETTERS,61(26),5.
MLA	Li, Xiaowei,et al."AcOH-mediated aerobic oxidative synthesis of 2-thioalkylbenzothiazoles via a three-component reaction".TETRAHEDRON LETTERS 61.26(2020):5.

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文件名称/大小	文献类型	版本类型	开放类型	使用许可
1-s2.0-S004040392030（819KB）	期刊论文	出版稿	限制开放	CC BY-NC-SA	浏览